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API Intermediates

API Intermediates

API intermediates are the essential chemical compounds formed during the synthesis of Active Pharmaceutical Ingredients (APIs). These intermediates play a critical role in defining the purity, efficacy, and overall quality of the final pharmaceutical product. Produced under strict regulatory compliance, API intermediates must meet rigorous quality standards to ensure they are safe and effective for further formulation.

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API Intermediates Products
SL NO. NAME OF THE PRODUCT CAS NO. API
1 2-Butylbenzofuran 4265-27-4 Amiodarone
2 5-Chlorovaleryl Chloride 1575-61-7 Apixaban
3 3,3-Dichloro-1-(4-nitrophenyl) piperidin-2-one 881386-01-2 Apixaban
4 3-Chloro-1-(4-nitrophenyl)-5,6-dihydropyridin-2(1H)-one 536760-29-9 Apixaban
5 5-Bromovaleryl Chloride 4509-90-4 Apixaban
6 3-Morpholino-1-(4-(2-oxopiperidin-1-yl)phenyl)-5,6-dihydropyridin-2(1H)-one 545445-44-1 Apixaban
7 2-Chloro-5-Iodobenzoic Acid 19094-56-5 Empagliflozin / Bexagliflozin / Dapagliflozin / Sotagliflozin
8 (2-Chloro-5-iodophenyl)(4-fluorophenyl) methanone 915095-86-2 Empagliflozin
9 (S)-(+)-3-Hydroxytetrahydrofuran 86087-23-2 Empagliflozin
10 5-Bromo-2-Chlorobenzoic Acid 21739-92-4 Dapagliflozin / Empagliflozin
11 (5-Bromo-2-chlorophenyl)(4-ethoxyphenyl) methanone 461432-22-4 Dapagliflozin / Sotagliflozin
12 5-Bromo-2-chloro-4-ethoxydiphenylmethane 461432-23-5 Dapagliflozin / Sotagliflozin
13 5-Iodo-2-chloro-4’-ethoxydiphenylmethanone 1103738-26-6 Dapagliflozin
14 5-Iodo-2-chloro-4’-ethoxydiphenylmethane 1103738-29-9 Dapagliflozin
15 2-Methyl-5-Iodobenzoic Acid 54811-38-0 Canagliflozin
16 L-Threonine Methyl Ester HCl 39994-75-7 Insulin
17 Iodobenzene 591-50-4 Pirfenidone
18 Chloroiodomethane 593-71-5 Vaniprevir
19 Diiodomethane 75-11-6 Etravirine
20 1-Bromo-2-iodobenzene 583-55-1 Vortioxetine
15 4-(4-Aminophenyl)morpholin-3-one 438056-69-0 Rivaroxaban
API Intermediates - Under Scale Up Products
SL NO. NAME OF THE PRODUCT CAS NO. API
1 p-Toluenesulfonylmethyl Isocyanide 36635-61-7 Bempedoic Acid
2 (3S)-3-[4-[(2-Chloro-5-iodophenyl) methyl] phenoxy] tetrahydro-furan 915095-94-2 Empagliflozin
3 S)-3-(4-(5-Bromo-2-chlorobenzyl)phenoxy)tetrahydrofuran 915095-89-5 Empagliflozin
4 2,3,4,6-Tetrakis-O-trimethylsilyl-D-gluconolactone 32384-65-9 Dapagliflozin / Empagliflozin
5 6-Nitro-1H-indazole 7597-18-4 -
6 4-iodobenzonitrile 3058-39-7 -
API Intermediates - Under Development Products
SL NO. NAME OF THE PRODUCT CAS NO. API
1 4-Bromo-2-Chlorobenzonitrile 154607-01-9 Darolutamide
2 Ethyl-7-Bromo-2,2-Dimethylheptanoate 123469-92-1 Bempedoic Acid
3 2,2,14,14-tetramethyl-8-oxopentadecaenedioic 413624-71-2 Bempedoic Acid
4 6-Iodo-1H-Indazole 261953-36-0 Axitinib
5 3-iodo-6-nitro-1-(tetrahydro-2-Hpyran-2-yl)-1H-indazole 886230-74-6 Axitinib
6 (E)-6-Iodo-3-[2-(pyridin-2-yl)ethenyl]-1-(tetrahydro-2H-pyran-2-yl)-1H-indazole 886230-77-9 Axitinib
7 2,3,4,6-Tetra-O-Benzyl-D-Glucopyranose 4132-28-9 Miglustat
8 3-(piperidin-4-yl)quinolin-2(1h)-one hydrochloride 855778-84-6 Zavegepant
9 1-(1-Methylpiperidin-4-yl)piperazine trihydrochloride 349535-15-5 Zavegepant
10 1-(1-Methylpiperidin-4-yl)piperazine 23995-88-2 Zavegepant
11 (2R,3R,4R,5S,6S)-2-(acetoxymethyl)-6-(4-chloro-3-(4-(((S)-tetrahydrofuran-3-yl)oxy)benzyl)phenyl) tetrahydro-2H-pyran-3,4,5-triyl triacetate 915095-99-7 Empagliflozin
12 2-Chloro-3-iodo-4-pyridinamime 909036-46-0 -